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Retatrutide

LY3437943, LY-3437943

A synthetic peptide acting as a triple agonist for GLP-1, GIP, and glucagon receptors, designed for treating obesity and type 2 diabetes by promoting weight loss and glycemic control.

Quick Stats
Studies 83
Trials 32
Formula C221H342N46O68
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Utility 4
pubmed Apr 1, 2025

Efficacy of GLP-1 Receptor Agonist-Based Therapies on Cardiovascular Events and Cardiometabolic Parameters in Obese Individuals Without Diabetes: A Meta-Analysis of Randomized Controlled Trials.

Yin. Yue Y; Zhang. Minghan M; Cao. Qiuyu Q; Lin. Lin L; Lu. Jieli J; Bi. Yufang Y; Chen. Yuhong Y

A big review of 29 trials found that drugs that act like GLP‑1 (including the newer peptide retatrutide) cut heart‑related events and improve blood pressure, weight, cholesterol and inflammation in overweight people who don’t have diabetes. This means you can get heart‑health and weight‑loss benefits from these drugs even if you’re not diabetic.

Utility 4
pubmed Jul 28, 2025

Triple Agonism Based Therapies for Obesity.

Goldney. Jonathan J; Hamza. Malak M; Surti. Farhaana F; Davies. Melanie J MJ; Papamargaritis. Dimitr...

Retatrutide is a new triple‑agonist drug that hits GLP‑1, GIP, and glucagon receptors. In early trials it caused massive weight loss – up to 24% in people with obesity and about 17% in those with type‑2 diabetes – and dramatically lowered blood sugar, blood pressure, cholesterol, waist size, and liver fat. The main side effects were typical gut upset, and no serious safety issues showed up yet.

Utility 4
pubmed Feb 17, 2024

A review of an investigational drug retatrutide, a novel triple agonist agent for the treatment of obesity.

Kaur. Manmeet M; Misra. Saurav S

Retatrutide is a new peptide that hits three hormone receptors (GLP‑1, GIP, and glucagon) and has shown big weight‑loss numbers in early trials – about 17% loss after 6 months and 24% after a year – while also being studied for diabetes and fatty liver. It’s still in Phase III, so it isn’t on the market yet, but the early data suggest it could become a powerful tool for cutting fat and improving metabolic health.

Utility 4
pubmed Nov 22, 2023

Advances in obesity pharmacotherapy; learning from metabolic surgery and beyond.

Tsilingiris. Dimitrios D; Kokkinos. Alexander A

The paper explains that the biggest weight‑loss success comes from bariatric surgery, which works partly by changing gut hormones. New drugs that combine GLP‑1, GIP, and glucagon signals (like retatrutide) can cause weight loss almost as big as surgery, opening the door to a non‑surgical "medical bypass" for obesity and related health problems.

Utility 4
pubmed Jun 26, 2023

Triple-Hormone-Receptor Agonist Retatrutide for Obesity - A Phase 2 Trial.

Jastreboff. Ania M AM; Kaplan. Lee M LM; Frías. Juan P JP; Wu. Qiwei Q; Du. Yu Y; Gurbuz. Sirel...

In a 48‑week trial, the triple‑hormone peptide retatrutide helped people with obesity lose a lot of weight – up to about 24% of body weight at the highest dose. The weight loss got bigger with higher doses, and most people on the 4‑8‑12 mg doses lost at least 10% of their weight. The main side effects were stomach‑related issues that got milder when the dose started lower, and there was a temporary rise in heart rate.

Utility 4
pubmed Jun 26, 2023

Retatrutide, a GIP, GLP-1 and glucagon receptor agonist, for people with type 2 diabetes: a randomised, double-blind, placebo and active-controlled, parallel-group, phase 2 trial conducted in the USA.

Rosenstock. Julio J; Frias. Juan J; Jastreboff. Ania M AM; Du. Yu Y; Lou. Jitong J; Gurbuz. Sirel S;...

In a phase‑2 trial, the experimental peptide retatrutide (which hits GIP, GLP‑1 and glucagon receptors) lowered blood sugar by up to 2 % and cut body weight by about 17 % after 36 weeks in people with type‑2 diabetes. The biggest effects were seen at the higher doses (8‑12 mg), and side‑effects were mainly mild stomach upset, similar to other GLP‑1 drugs.

Utility 4
pubmed Jul 29, 2025

Glucagon-like peptide-1 receptor analogues and beyond: emerging obesity pharmacotherapies.

Abburi. Kaivalya K; Melson. Eka E; Miras. Alexander D AD; Papamargaritis. Dimitris D

A new drug combo called retatrutide, which hits three gut hormones (GLP‑1, GIP, and glucagon), is showing weight‑loss results that are almost as good as bariatric surgery. This is part of a wave of next‑generation obesity pills that go beyond the single‑hormone drugs we already have.

Utility 4
pubmed Apr 16, 2025

Antiobesity medications in adult and pediatric obesity and metabolic dysfunction-associated steatotic liver disease.

Rodriguez. Natalie N; Hartmann. Phillipp P

Retatrutide, a new anti‑obesity peptide, cut body weight by about 22% compared with placebo and slashed liver fat by roughly 80% in adult trials lasting 48‑72 weeks. It performed even better than other popular drugs like semaglutide and tirzepatide, showing strong promise for tackling obesity and fatty‑liver disease.

Utility 4
pubmed Jan 7, 2025

Efficacy and Safety of Glucagon-Like Peptide-1 Receptor Agonists for Weight Loss Among Adults Without Diabetes : A Systematic Review of Randomized Controlled Trials.

Moiz. Areesha A; Filion. Kristian B KB; Toutounchi. Helia H; Tsoukas. Michael A MA; Yu. Oriana H Y O...

A review of recent trials shows that the experimental peptide retatrutide can cut body weight by about 22% after roughly a year of weekly injections, outperforming other GLP‑1 drugs like semaglutide and tirzepatide. Most side effects are stomach‑related (nausea, vomiting, diarrhea) and usually mild, though a few people stopped treatment because of them.

Utility 4
pubmed Oct 30, 2024

The impact of weight loss on fat-free mass, muscle, bone and hematopoiesis health: Implications for emerging pharmacotherapies aiming at fat reduction and lean mass preservation.

Stefanakis. Konstantinos K; Kokkorakis. Michail M; Mantzoros. Christos S CS

Big weight‑loss drugs like tirzepatide (and the newer retatrutide) can drop 15‑25% of body weight, but about a quarter of that loss is muscle and bone, which can hurt health, especially as you age. New drugs that block myostatin/activin (e.g., Bimagrumab, Trevogrumab, Garetosmab) may help keep muscle and bone while you lose fat, and combining them with incretin agonists could give a better body‑composition outcome.

Utility 4
pubmed Feb 14, 2024

The Road towards Triple Agonists: Glucagon-Like Peptide 1, Glucose-Dependent Insulinotropic Polypeptide and Glucagon Receptor - An Update.

Jakubowska. Agnieszka A; Roux. Carel W le CWL; Viljoen. Adie A

A recent phase‑2 trial tested retatrutide, a drug that hits three gut hormone receptors (GLP‑1, GIP, and glucagon). Over 48 weeks, participants taking the highest dose (12 mg) lost about 24% of their body weight, while also seeing improvements in blood sugar, cholesterol, blood pressure, inflammation, and liver fat. The study shows that hitting all three pathways at once can produce very strong weight‑loss results.

Utility 3
pubmed Sep 13, 2024

Effects of once-weekly subcutaneous retatrutide on weight and metabolic markers: A systematic review and meta-analysis of randomized controlled trials.

Pasqualotto. Eric E; Ferreira. Rafael Oliva Morgado ROM; Chavez. Matheus Pedrotti MP; Hohl. Alexandr...

A review of three clinical trials found that once‑weekly injections of retatrutide can cut body weight by about 10 kg (roughly 10% of body weight) and improve BMI and waist size in people who are overweight, obese, or have type‑2 diabetes. A lot more people on the drug hit big weight‑loss milestones (5%, 10%, 15% and even 20% loss) compared with placebo, though mild stomach upset and allergic‑type reactions were a bit more common.

Utility 3
pubmed Nov 7, 2023

Enteroendocrine cell regulation of the gut-brain axis.

Barton. Joshua R JR; Londregan. Annie K AK; Alexander. Tyler D TD; Entezari. Ariana A AA; Covarrubia...

This review explains how gut hormone‑producing cells (EECs) talk to the brain, and why drugs like semaglutide, terzepatide and the experimental peptide retatrutide work for weight loss and diabetes. It highlights that some EECs can send fast signals directly to nerves, and that understanding these pathways could help create better treatments for obesity and gut disorders.

Utility 3
pubmed May 30, 2025

Retatrutide-A Game Changer in Obesity Pharmacotherapy.

Katsi. Vasiliki V; Koutsopoulos. Georgios G; Fragoulis. Christos C; Dimitriadis. Kyriakos K; Tsioufi...

Retatrutide is a new drug that hits three hormone receptors (GLP‑1, GIP, and glucagon) at once. Early animal work and Phase I‑II trials show it can cut body weight, lower blood sugar, and improve liver and kidney health, but it mainly causes stomach‑related side effects and is still being tested in larger Phase III studies.

Utility 3
pubmed Oct 19, 2024

The "Weight" for a New Agent Is Almost Over: A Commentary on the Novel Triagonist Retatrutide for Obesity.

Deravi. Maryam M; Piszczatoski. Chris C; Phillips. Bradley B; Huston. Jessica J; Vascimini. Angelina...

Retatrutide is a new drug that hits three hormone receptors (glucagon, GLP‑1, and GIP) and has shown in early trials that people can lose up to about a quarter of their body weight and shrink their waist by almost 20 cm, with the main side‑effects being stomach upset.

Utility 3
pubmed Aug 30, 2024

Comparison of the effects of Liraglutide, Tirzepatide, and Retatrutide on diabetic kidney disease in db/db mice.

Ma. Jun J; Hu. Xiaoyan X; Zhang. Wencheng W; Tao. Mengyuan M; Wang. Min M; Lu. Weiping W

In a mouse study, the experimental drug retatrutide helped the animals lose more weight and protect their kidneys better than the already‑approved drugs liraglutide and tirzepatide. It also improved liver health, lowered bad cholesterol, raised good cholesterol, and boosted a gut‑derived molecule (butyrate) linked to a healthier microbiome. However, retatrutide wasn’t any better than tirzepatide at lowering blood sugar.

Utility 3
pubmed Jan 23, 2024

Future is Brighter: New Potential Paradigm-Shifting Medications and Regimens for Diabetes and Obesity.

Al-Horani. Rami A RA; Aliter. Kholoud F KF; Aliter. Hashem F HF

The abstract reviews new drugs for diabetes and obesity, highlighting retatrutide as one of several promising treatments that could dramatically improve blood sugar control and weight loss. While it doesn’t give dosing details, it signals that retatrutide is moving through advanced trials and may become a powerful tool for people looking to manage metabolic health.

Utility 3
pubmed Nov 6, 2024

The power of three: Retatrutide's role in modern obesity and diabetes therapy.

Abdul-Rahman. Toufik T; Roy. Poulami P; Ahmed. Fatma Kamal FK; Mueller-Gomez. Jann Ludwig JL; Sarkar...

Retatrutide is a new drug that hits three gut hormone receptors at once, helping people lose weight, lower blood sugar, and possibly improve heart health. Early trials (phases 1‑3) show big drops in body weight and better glucose control, but we still need more data on long‑term safety and how it works in special groups like kids.

Utility 3
pubmed Mar 14, 2025

Incretin triple agonist retatrutide (LY3437943) alleviates obesity-associated cancer progression.

Marathe. Sandesh J SJ; Grey. Emily W EW; Bohm. Margaret S MS; Joseph. Sydney C SC; Ramesh. Arvind V...

In mouse studies, the weight‑loss drug retatrutide not only shrank body fat but also dramatically slowed the growth of pancreatic and lung cancers linked to obesity. Even after the drug was stopped, the anti‑cancer effects stuck around, likely because it reshaped the immune system to be more anti‑tumor.

Utility 3
pubmed Jul 4, 2025

Inotropic effects of retatrutide in isolated human atrial preparations.

Neumann. Joachim J; Ahlrep. Undine U; Hofmann. Britt B; Gergs. Ulrich U

The study shows that retatrutide, a drug being developed for diabetes and obesity, can make human heart muscle cells contract stronger and relax faster in lab experiments. This effect comes from activating several hormone receptors that raise cAMP levels inside the cells. The findings are based on heart tissue taken from patients with severe coronary disease, not on healthy volunteers or real‑world use.