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Sermorelin

GHRH (1-29), GRF 1-29 NH2, Sermorelin acetate

A synthetic 29-amino acid analog of growth hormone-releasing hormone that stimulates pituitary gland to release growth hormone.

Quick Stats
Studies 223
Trials 41
Formula C149H246N44O42S
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Utility 2
pubmed 1987

Injection of synthetic human growth hormone-releasing factors in dairy cows. 1. Effect on feed intake and milk yield and composition.

Pelletier. G G; Petitclerc. D D; Lapierre. H H; Bernier-Cardou. M M; Morisset. J J; Gaudreau. P P; C...

In a study with dairy cows, giving synthetic human growth hormone‑releasing factor (either the full 44‑amino‑acid version or a shorter 29‑amino‑acid fragment) boosted milk production by about 15‑19% without changing how much the cows ate, and it made the feed they did eat work more efficiently.

Utility 2
pubmed Mar 16, 1999

Inhibition of growth, production of insulin-like growth factor-II (IGF-II), and expression of IGF-II mRNA of human cancer cell lines by antagonistic analogs of growth hormone-releasing hormone in vitro.

Csernus. V J VJ; Schally. A V AV; Kiaris. H H; Armatis. P P

The study shows that chemicals that block the hormone that normally tells the pituitary to release growth hormone (called GHRH antagonists) can slow the growth of several cancer cell lines by cutting down the amount of a growth factor called IGF‑II that many tumors make themselves. This effect is separate from the usual growth‑hormone/IGF‑I pathway and works by interfering with the tumor’s own IGF‑II signaling loop.

Utility 2
pubmed Oct 1, 1990

Characterization of [125I-Tyr10]human growth hormone-releasing factor (1-44) amide binding to rat pituitary: evidence for high and low affinity classes of sites.

Abribat. T T; Boulanger. L L; Gaudreau. P P

Researchers measured how a radioactive version of human growth hormone‑releasing factor (GRF, also called sermorelin) sticks to rat pituitary tissue. They found two kinds of binding spots: one that grabs the peptide tightly but in small numbers, and another that holds it more loosely but in larger numbers. The test works best with a modest amount of magnesium, and the binding can be stopped with EDTA to keep the peptide stable.

Utility 2
pubmed 1990

The plasma pattern of growth hormone in conscious rats during late pregnancy.

Carlsson. L L; Edén. S S; Jansson. J O JO

In pregnant rats, blood levels of growth hormone (GH) rise a lot during the later stages of pregnancy, especially on day 20, mainly because the baseline GH goes up and the bursts of GH become larger. Giving a human GH‑releasing factor (GRF) analogue still boosts GH, but if the pituitary gland is removed, GH disappears, showing the pituitary is the source.

Utility 2
pubmed 1991

Influence of growth hormone-releasing hormone (GHRH) on phytohemagglutinin-induced lymphocyte activation: comparison of two synthetic forms. GHRH and PHA-induced lymphocyte activation.

Valtorta. A A; Moretta. A A; Maccario. R R; Bozzola. M M; Severi. F F

In a lab test, tiny amounts of the short form of human growth‑hormone‑releasing hormone (GHRH 1‑29) helped immune cells multiply when they were stimulated, but larger amounts actually slowed their activity and reduced a key immune signal (IL‑2). The longer form (GHRH 1‑44) didn’t change anything, and the hormone wasn’t toxic to the cells.

Utility 2
pubmed 1985

Effect of different growth hormone-releasing factors on the concentrations of growth hormone, insulin and metabolites in the plasma of sheep maintained in positive and negative energy balance.

Hart. I C IC; Chadwick. P M PM; Coert. A A; James. S S; Simmonds. A D AD

In sheep, different forms of growth‑hormone‑releasing factor (including ones similar to sermorelin) all boosted GH levels, and the boost was actually bigger when the animals were on a restricted diet. The type of GRF mattered less than whether the animal was eating a lot or a little.

Utility 2
pubmed Feb 29, 1984

Super-active analogs of growth hormone-releasing factor (1-29)-amide.

Lance. V A VA; Murphy. W A WA; Sueiras-Diaz. J J; Coy. D H DH

Scientists made several modified versions of the growth‑hormone‑releasing peptide (like sermorelin) and tested them in rats and pigs. One version, with a D‑alanine at position 2, was about 50 times stronger at making the body release growth hormone than the regular peptide. The other tweaks were also stronger than the original, but not as dramatic.

Utility 1
pubmed Oct 17, 2024

A novel approach for the treatment of AML, through GHRH antagonism: MIA-602.

Costoya. Joel J; Gaumond. Simonetta I SI; Chale. Ravinder S RS; Schally. Andrew V AV; Jimenez. Joaqu...

The study looks at a new drug called MIA-602 that blocks a hormone signal (GHRH) and shows it can kill leukemia cells in lab tests, even those that resist standard chemo, and works better when combined with chemo. However, this is early‑stage cancer research, not a health‑boosting supplement, and it isn’t ready for personal use.

Utility 1
pubmed Apr 1, 2025

Growth Hormone-Releasing Hormone Antagonists Increase Radiosensitivity in Non-Small Cell Lung Cancer Cells.

Gesmundo. Iacopo I; Pedrolli. Francesca F; Giglioli. Francesca Romana FR; Jazaj. Florian F; Granato....

Scientists found that drugs that block the hormone that normally tells the body to release growth hormone can make lung cancer cells more vulnerable to radiation in lab dishes, but this research used special lab compounds, not the growth‑hormone‑releasing peptide sermorelin, and it’s far from any real‑world self‑experiment or treatment plan.

Utility 1
pubmed Jun 6, 2011

Effects of the growth hormone-releasing hormone (GH-RH) antagonist on brain functions in mice.

Telegdy. Gyula G; Tanaka. Masaru M; Schally. Andrew V AV

In mice, a brain‑injected GH‑releasing hormone blocker called MZ‑4‑71 helped them remember a task better, stopped memory loss caused by a beta‑amyloid peptide, and showed mild anti‑depression and anti‑anxiety effects, without changing general activity. However, the study used direct brain injections in animals, so it doesn’t give clear guidance for people to use this or related peptides like sermorelin in real life.

Utility 1
pubmed Oct 3, 2009

GHRH antagonist causes DNA damage leading to p21 mediated cell cycle arrest and apoptosis in human colon cancer cells.

Hohla. Florian F; Buchholz. Stefan S; Schally. Andrew V AV; Seitz. Stefan S; Rick. Ferenc G FG; Szal...

The study shows that a synthetic molecule that blocks growth‑hormone‑releasing hormone (GHRH) can damage DNA in colon‑cancer cells, trigger cell‑death pathways, and shrink tumors in mice, but it doesn’t tell you how to use it for health‑boosting or longevity in normal people.

Utility 1
pubmed Mar 2, 2020

Signaling mechanisms of growth hormone-releasing hormone receptor in LPS-induced acute ocular inflammation.

Liang. Wei Cheng WC; Ren. Jia Lin JL; Yu. Qiu Xiao QX; Li. Jian J; Ng. Tsz Kin TK; Chu. Wai Kit WK;...

The study shows that the receptor for growth‑hormone‑releasing hormone (GHRH‑R) helps drive eye inflammation by activating a JAK2‑STAT3 signaling chain, and that blocking this receptor or using a JAK inhibitor can calm the inflammation in animal and cell models.

Utility 1
pubmed Feb 17, 2012

Combining growth hormone-releasing hormone antagonist with luteinizing hormone-releasing hormone antagonist greatly augments benign prostatic hyperplasia shrinkage.

Rick. Ferenc G FG; Szalontay. Luca L; Schally. Andrew V AV; Block. Norman L NL; Nadji. Mehrdad M; Sz...

In rats with hormone‑induced enlarged prostates, giving a drug that blocks growth‑hormone‑releasing hormone (GHRH) together with a drug that blocks luteinizing‑hormone‑releasing hormone (LHRH) cut prostate size by about 30% and lowered several prostate‑related blood markers.

Utility 1
pubmed Feb 14, 2011

Antagonists of growth hormone-releasing hormone (GHRH) reduce prostate size in experimental benign prostatic hyperplasia.

Rick. Ferenc G FG; Schally. Andrew V AV; Block. Norman L NL; Nadji. Mehrdad M; Szepeshazi. Karoly K;...

In a rat study, drugs that block the hormone GHRH shrank enlarged prostates by about 18‑21% after six weeks and lowered inflammation markers, but the work used GHRH antagonists, not the growth‑stimulating peptide sermorelin, and was done only in animals.

Utility 1
pubmed Jul 27, 2011

Inhibitory effects of antagonists of growth hormone releasing hormone on experimental prostate cancers are associated with upregulation of wild-type p53 and decrease in p21 and mutant p53 proteins.

Stangelberger. Anton A; Schally. Andrew V AV; Rick. Ferenc G FG; Varga. Jozsef L JL; Baker. Benjamin...

In mouse studies, a drug that blocks the growth‑hormone‑releasing hormone (GHRH) slowed the growth of prostate cancer tumors and changed key cancer‑related proteins, especially p53. Adding another hormone blocker (Cetrorelix) made the effect stronger. The work doesn’t involve sermorelin (a GHRH‑activating peptide) and offers no direct guidance for human use.

Utility 1
pubmed Nov 1, 2011

GHRH antagonist MZ-5-156 increases the expression of AMPK in A549 lung cancer cells.

Siejka. Agnieszka A; Barabutis. Nektarios N; Schally. Andrew V AV

A lab study found that a synthetic growth‑hormone‑releasing‑hormone blocker (MZ‑5‑156) can slow the growth of lung cancer cells by turning on a cellular energy sensor called AMPK and shutting down growth signals, but this was only shown in cancer cells in a dish, not in people.

Utility 1
pubmed Jul 20, 2012

GHRH antagonist inhibits focal adhesion kinase (FAK) and decreases expression of vascular endothelial growth factor (VEGF) in human lung cancer cells in vitro.

Siejka. Agnieszka A; Barabutis. Nektarios N; Schally. Andrew V AV

The study found that a lab-made GHRH blocker (MZ-5-156) can shut down a signaling protein (FAK) and lower levels of molecules that help lung cancer cells grow new blood vessels and invade tissue, but this was only shown in cell dishes and uses a compound not available to the public.

Utility 1
pubmed Oct 24, 2012

GHRH antagonist when combined with cytotoxic agents induces S-phase arrest and additive growth inhibition of human colon cancer.

Rick. Ferenc G FG; Seitz. Stephan S; Schally. Andrew V AV; Szalontay. Luca L; Krishan. Awtar A; Datz...

A study found that a growth‑hormone‑releasing‑hormone blocker called JMR‑132 can pause colon‑cancer cells in the DNA‑making phase and make chemotherapy work better in lab dishes and mice, shrinking tumors by up to half. This isn’t about sermorelin (a hormone‑boosting peptide) and it’s only in animals, so it doesn’t give a usable plan for everyday health hacking.

Utility 1
pubmed Jul 27, 2012

Inhibitory effects of antagonists of growth hormone-releasing hormone on growth and invasiveness of PC3 human prostate cancer.

Muñoz-Moreno. Laura L; Arenas. M Isabel MI; Schally. Andrew V AV; Fernández-Martínez....

This study tested two chemicals that block the hormone that normally tells the body to release growth hormone. In mice with aggressive prostate cancer, these blockers slowed tumor growth and reduced markers linked to blood‑vessel formation and spread. The work is about cancer treatment, not about using growth‑hormone‑releasing peptides like sermorelin for health‑boosting purposes.