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Kisspeptin-10

KP-10, Metastin (45-54), Kisspeptin-10 (human), KiSS-1

Kisspeptin-10 is a decapeptide that activates the KISS1R receptor to stimulate GnRH release, regulating the reproductive hormone axis and fertility.

Quick Stats
Studies 877
Trials 47
Formula C63H83N17O14
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Utility 2
pubmed Apr 2, 2010

The role of kisspeptin signalling in the regulation of the GnRH-gonadotrophin ovarian axis in mice.

Colledge. W H WH; d'Anglemont de Tassigny. X X

This study shows that kisspeptin, a small protein made from the Kiss1 gene, is crucial for turning on the brain‑pituitary‑ovary hormone system that drives puberty and ovulation in mice. If the kisspeptin pathway is broken, animals (and humans) don’t develop normally and become infertile. The researchers also think kisspeptin might act directly in the ovary and placenta, not just in the brain.

Utility 2
pubmed Jan 31, 2005

Increased hypothalamic GPR54 signaling: a potential mechanism for initiation of puberty in primates.

Shahab. Muhammad M; Mastronardi. Claudio C; Seminara. Stephanie B SB; Crowley. William F WF; Ojeda....

In young monkeys, giving the peptide kisspeptin‑10 directly into the brain or bloodstream caused a strong release of the hormone GnRH, which then boosted luteinizing hormone (LH). The study also showed that the genes for kisspeptin (KiSS‑1) and its receptor (GPR54) become more active as the animals approach puberty, especially in females. This suggests that kisspeptin signaling helps kick‑start puberty by turning on the brain’s GnRH system.

Utility 2
pubmed Jun 24, 2004

A role for kisspeptins in the regulation of gonadotropin secretion in the mouse.

Gottsch. M L ML; Cunningham. M J MJ; Smith. J T JT; Popa. S M SM; Acohido. B V BV; Crowley. W F WF;...

In mice, giving kisspeptin peptides straight into the brain makes the pituitary release more LH (and at higher doses also FSH), showing that kisspeptin can turn on the reproductive hormone system, but the study used tiny brain injections that aren’t doable in people.

Utility 2
pubmed Aug 29, 2006

KiSS-1 and reproduction: focus on its role in the metabolic regulation of fertility.

Tena-Sempere. Manuel M

Kisspeptin, a brain chemical made by the KiSS-1 gene, is a key switch for starting puberty and keeping the reproductive hormone system running. When the body is low on energy (like during dieting or illness), kisspeptin levels fall, which can shut down fertility. Giving extra kisspeptin or boosting leptin (the fat‑cell hormone) can reverse this shutdown in animal studies, suggesting a link between energy balance and reproductive health.

Utility 2
pubmed Mar 23, 2007

Kisspeptin: a key link to seasonal breeding.

Revel. Florent G FG; Ansel. Laura L; Klosen. Paul P; Saboureau. Michel M; Pévet. Paul P; Mikkel...

The study shows that in hamsters, the hormone melatonin controls a brain signal called kisspeptin, which in turn drives the reproductive system. When day length is short, melatonin lowers kisspeptin levels and suppresses fertility, but giving extra kisspeptin can jump‑start testicular activity even in those conditions. This reveals a link between light cycles, melatonin, and reproductive hormones, but it’s based on animal experiments and doesn’t give direct guidance for human use.

Utility 2
pubmed Dec 25, 2008

Kisspeptins and GnRH neuronal signalling.

Colledge. William H WH

Kisspeptin is a small protein that talks to the brain cells that control reproductive hormones. When it binds to its receptor on GnRH neurons, it makes those cells fire more, releasing more GnRH and turning on the whole reproductive hormone system. The review explains how this signaling works at the cellular level across different animals.

Utility 2
pubmed Jun 8, 2006

Kisspepeptin-GPR54 signaling in the neuroendocrine reproductive axis.

Gottsch. M L ML; Clifton. D K DK; Steiner. R A RA

Kisspeptin is a brain chemical that tells the hormone-releasing system to start making reproductive hormones, and its partner receptor GPR54 is essential for puberty and fertility. If this system is broken, people can have very low sex hormones. The review explains how kisspeptin neurons react to the body’s own sex hormones, acting as a feedback loop.

Utility 2
pubmed Jul 3, 2008

Reproductive functions of kisspeptin and Gpr54 across the life cycle of mice and men.

Chan. Yee-Ming YM; Broder-Fingert. Sarabeth S; Seminara. Stephanie B SB

The study shows that the kisspeptin protein and its receptor GPR54 are essential for the brain's control of reproductive hormones throughout life. When either is broken by genetic mutations, people and mice can have anything from mild to severe underdevelopment of sexual characteristics. In short, kisspeptin acts like a messenger that tells the hormone‑releasing system when to turn on.

Utility 2
pubmed Apr 18, 2006

Kisspeptin immunoreactive cells of the ovine preoptic area and arcuate nucleus co-express estrogen receptor alpha.

Franceschini. I I; Lomet. D D; Cateau. M M; Delsol. G G; Tillet. Y Y; Caraty. A A

Researchers found that in sheep brains, cells that make the hormone‑like peptide kisspeptin‑10 also have estrogen receptors, especially in areas that control reproductive hormones. This suggests kisspeptin works together with estrogen to regulate the release of GnRH and LH, which are key for fertility.

Utility 2
pubmed Mar 2, 2006

Effects of single or repeated intravenous administration of kisspeptin upon dynamic LH secretion in conscious male rats.

Tovar. S S; Vázquez. M J MJ; Navarro. V M VM; Fernández-Fernández. R R; Castellano. J...

In awake male rats, tiny IV doses of the peptide kisspeptin-10 quickly trigger strong bursts of the hormone LH, which controls reproductive function. The effect works even when the rats are fasting, and giving the peptide repeatedly keeps the LH spikes steady. A longer version of the peptide (kisspeptin-52) does the same thing but a bit stronger.

Utility 2
pubmed May 30, 2008

Kisspeptin and KISS1R: a critical pathway in the reproductive system.

Gianetti. Elena E; Seminara. Stephanie S

The paper explains that kisspeptin and its receptor KISS1R are crucial switches that start puberty and control reproductive hormones. They help the brain release GnRH, which then triggers the release of sex hormones, and genetic changes in this system can cause delayed or early puberty.

Utility 2
pubmed Mar 9, 2006

Hypothalamic expression of KiSS-1 system and gonadotropin-releasing effects of kisspeptin in different reproductive states of the female Rat.

Roa. J J; Vigo. E E; Castellano. J M JM; Navarro. V M VM; Fernández-Fernández. R R; Casanu...

In adult female rats, a single brain injection of kisspeptin-10 reliably triggers bursts of the reproductive hormones LH and FSH. The response is strongest at estrus and even tiny doses work during diestrus. Removing the ovaries doesn’t stop the effect, but restoring estrogen and progesterone brings the hormone spikes back to full strength. During pregnancy and lactation, the rats still respond, with especially high sensitivity in pregnant females, and the brain’s kisspeptin gene (KiSS-1) is turned up.

Utility 2
pubmed Jan 6, 2007

GPR54 and KiSS-1: role in the regulation of puberty and reproduction.

Kuohung. Wendy W; Kaiser. Ursula B UB

This study shows that the kisspeptin‑GPR54 system is essential for starting puberty by activating the brain's GnRH neurons, which then trigger hormone release. While it explains how the pathway works, it doesn’t give any dosing or protocol details for everyday use.

Utility 2
pubmed Jun 8, 2006

Novel signals for the integration of energy balance and reproduction.

Fernandez-Fernandez. R R; Martini. A C AC; Navarro. V M VM; Castellano. J M JM; Dieguez. C C; Aguila...

The paper explains that the brain peptide kisspeptin helps link how much energy you have (like body weight and food intake) with your reproductive system. It works together with other gut hormones like ghrelin and PYY, and its levels drop when you’re in a calorie deficit, which can suppress fertility.

Utility 2
pubmed 2004

Central and peripheral administration of kisspeptin-10 stimulates the hypothalamic-pituitary-gonadal axis.

Thompson. E L EL; Patterson. M M; Murphy. K G KG; Smith. K L KL; Dhillo. W S WS; Todd. J F JF; Ghate...

In male rats, giving the short peptide kisspeptin-10 either directly into the brain or into the bloodstream quickly raised the hormones that control reproduction (LH, FSH) and boosted testosterone levels. The brain‑derived hormone that triggers LH release (LHRH) also went up, showing the effect works through the normal hypothalamic‑pituitary‑gonadal pathway.

Utility 2
pubmed Jun 1, 2006

Mechanisms of Disease: the first kiss-a crucial role for kisspeptin-1 and its receptor, G-protein-coupled receptor 54, in puberty and reproduction.

Seminara. Stephanie B SB

The paper explains that a protein called kisspeptin and its receptor GPR54 are key triggers for the hormone GnRH, which starts puberty and controls reproductive hormones. If the receptor doesn’t work (due to genetic mutations), puberty doesn’t happen. Giving kisspeptin fragments can strongly stimulate GnRH release, showing this pathway is a major driver of reproductive hormone signaling.

Utility 2
pubmed May 24, 2007

Laeverin/aminopeptidase Q, a novel bestatin-sensitive leucine aminopeptidase belonging to the M1 family of aminopeptidases.

Maruyama. Masato M; Hattori. Akira A; Goto. Yoshikuni Y; Ueda. Masamichi M; Maeda. Michiyuki M; Fuji...

Researchers discovered that a protein called Laeverin (also known as aminopeptidase Q) can cut the kisspeptin-10 peptide, which is important for hormone signaling. This enzyme works best on leucine‑containing sequences and is strongly blocked by the drug bestatin. The finding suggests that the body can break down kisspein‑10 in the placenta, and that bestatin could be used to slow that breakdown.

Utility 2
pubmed Sep 5, 2006

Kisspeptin mediates the photoperiodic control of reproduction in hamsters.

Revel. Florent G FG; Saboureau. Michel M; Masson-Pévet. Mireille M; Pévet. Paul P; Mikkels...

The study shows that the peptide kisspeptin-10 can jump‑start reproductive activity in hamsters that are normally suppressed by short daylight, and that this effect depends on melatonin signaling. In simple terms, giving kisspeptin-10 to these animals over time re‑activated their testes even when the environment would normally keep them inactive.