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Kisspeptin-10

KP-10, Metastin (45-54), Kisspeptin-10 (human), KiSS-1

Kisspeptin-10 is a decapeptide that activates the KISS1R receptor to stimulate GnRH release, regulating the reproductive hormone axis and fertility.

Quick Stats
Studies 877
Trials 47
Formula C63H83N17O14
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Utility 2
pubmed Oct 21, 2009

Regulation of GPR54 signaling by GRK2 and {beta}-arrestin.

Pampillo. Macarena M; Camuso. Natasha N; Taylor. Jay E JE; Szereszewski. Jacob M JM; Ahow. Maryse R...

The study shows that the kisspeptin receptor (GPR54) can become less responsive when it interacts with proteins called GRK2 and beta‑arrestin, and that these proteins also shape downstream signaling inside cells. This is basic cell‑biology work, not a human trial, but it hints that repeated kisspeptin use could lead to desensitization.

Utility 2
pubmed Aug 29, 2009

The recent genetics of hypogonadotrophic hypogonadism - novel insights and new questions.

Semple. Robert K RK; Topaloglu. A Kemal AK

This review explains that many genes can cause a condition where the brain doesn’t signal the gonads properly, leading to low sex hormones. Recent genetic work showed that the peptide kisspeptin is a key trigger for releasing the hormone GnRH, which starts the whole reproductive hormone cascade. While this confirms kisspein’s importance, the paper doesn’t give any dosing or practical tips for using kisspeptin-10 in everyday health hacks.

Utility 2
pubmed Apr 6, 2011

Kisspeptin resets the hypothalamic GnRH clock in men.

Chan. Yee-Ming YM; Butler. James P JP; Pinnell. Nancy E NE; Pralong. François P FP; Crowley. Wi...

Giving men a single IV dose of the short kisspeptin peptide (kisspeptin-10) caused a quick, strong surge in the hormone LH, which reflects GnRH activity. This surge was bigger than the body’s normal pulses and lasted about 17 minutes, and it also pushed back the timing of the next natural pulse, effectively resetting the hormone clock.

Utility 2
pubmed Sep 29, 2009

Characteristics of the stimulatory effect of kisspeptin-10 on the secretion of luteinizing hormone, follicle-stimulating hormone and growth hormone in prepubertal male and female cattle.

Ezzat Ahmed. Ahmed A; Saito. Hayato H; Sawada. Tatsuru T; Yaegashi. Tomoyoshi T; Yamashita. Tetsuro...

In a small study on young cattle, giving the peptide kisspeptin‑10 caused a quick rise in the reproductive hormones LH and FSH, especially when injected into a vein and more strongly in male calves. It didn’t change growth hormone levels, and an intramuscular shot worked but not as well as the IV dose.

Utility 2
pubmed Jul 30, 2010

Why kisspeptin is such important for reproduction?

Meczekalski. Blazej B; Podfigurna-Stopa. Agnieszka A; Genazzani. Andrea Riccardo AR

Kisspeptin is a brain chemical that helps turn on the hormone chain that controls puberty, fertility, and the menstrual cycle. It works mainly in the hypothalamus but also affects the pituitary and ovaries, and its levels drop when the body is low on energy. Mutations that block its receptor cause delayed puberty, while over‑active signaling can lead to early puberty. Researchers think kisspeptin could someday be used to tweak the reproductive hormone system or even treat some cancers, but more work is needed.

Utility 2
pubmed Nov 1, 2010

The effects of kisspeptin-54 on blood pressure in humans and plasma kisspeptin concentrations in hypertensive diseases of pregnancy.

Nijher. Gurjinder M K GM; Chaudhri. Owais B OB; Ramachandran. Radha R; Murphy. Kevin G KG; Zac-Vargh...

Giving kisspeptin-54 to healthy men and women didn't change their heart rate or blood pressure, and the amount of kisspeptin naturally circulating in pregnant women didn't predict blood pressure or differ between normal and hypertensive pregnancies.

Utility 2
pubmed Apr 2, 2010

Kisspeptins and the metabolic control of reproduction: physiologic roles and physiopathological implications.

Tena-Sempere. M M

Researchers found that a brain peptide called kisspeptin helps connect the body’s energy status to the hormones that control reproduction. In mice, kisspeptin neurons receive signals like leptin (a fat‑derived hormone) and pass them on to GnRH, the master hormone for fertility, possibly using the Crtc1 and mTOR pathways. This shows a direct link between metabolism and reproductive health, but the work is still early and in animals only.

Utility 2
pubmed Apr 8, 2010

Role of kisspeptin/GPR54 system in human reproductive axis.

Silveira. Leticia F G LFG; Teles. Milena G MG; Trarbach. Ericka B EB; Latronico. Ana Claudia AC

Kisspeptin is a protein that acts like a switch to turn on the brain’s hormone system that controls puberty and reproduction. It boosts the release of hormones that tell the gonads to make sex hormones, and its levels rise during puberty. Mutations that stop kisspeptin or its receptor from working cause delayed or absent puberty, showing how essential it is.

Utility 2
pubmed Apr 8, 2010

Biology of kisspeptins.

Hameed. Saira S; Dhillo. Waljit S WS

Kisspeptin is a brain chemical that acts like a switch for starting puberty and keeping the reproductive hormone system running smoothly. The review explains how this peptide works, why it matters for fertility, and how problems with its signaling can cause a condition where the body doesn’t produce enough sex hormones.

Utility 2
pubmed Mar 9, 2009

Molecular interaction between kisspeptin decapeptide analogs and a lipid membrane.

Lee. Ju Yeon JY; Moon. Jung Sun JS; Eu. Young-Jae YJ; Lee. Chul Won CW; Yang. Sung-Tae ST; Lee. Seun...

The study shows that kisspein-10 needs to stick to cell membranes to work well, and tiny changes to its structure can stop it from activating its receptor. The peptide folds into tight turns rather than helices when near membranes, suggesting it may travel with the membrane to reach its target.

Utility 2
pubmed Nov 7, 2009

Presence of kisspeptin-like immunoreactivity in human adrenal glands and adrenal tumors.

Takahashi. Kazuhiro K; Shoji. Itaru I; Shibasaki. Akiko A; Kato. Ichiro I; Hiraishi. Keisuke K; Yama...

Scientists discovered that the hormone‑like peptide kisspeptin is naturally present in human adrenal glands and in various adrenal tumors, with similar amounts across normal tissue and different tumor types, and it’s especially strong in the adrenal medulla.

Utility 2
pubmed Jul 31, 2010

Kisspeptin: a critical regulator of puberty and reproductive function.

Sam. Amir H AH; Dhillo. Waljit S WS

Kisspein-10 is a protein that helps start puberty and control reproductive hormones by telling the brain to release GnRH, which then triggers gonadotropins. Mutations that stop its receptor cause low hormone levels, while activating mutations can cause early puberty. Scientists see it as a possible drug target for tweaking the reproductive hormone system, but there are no ready‑to‑use dosing guidelines yet.

Utility 2
pubmed 2010

Molecular causes of hypogonadotropic hypogonadism.

Topaloglu. Ali Kemal AK; Kotan. Leman Damla LD

The paper explains that puberty and reproductive hormone release are controlled by a complex network of genes and signals, including kisspeptin and neurokinin B. Only about a third of genetic cases of low gonadotropin levels are explained by known mutations, and many genes can interact, making the condition variable. While this deepens scientific understanding, it doesn’t give clear, ready‑to‑use instructions for using kisspeptin‑10 in health‑hacking protocols.

Utility 2
pubmed Mar 24, 2009

Nuclear magnetic resonance and circular dichroism study of metastin (Kisspeptin-54) structure in solution.

Shin. Ronald R; Welch. Danny R DR; Mishra. Vinod K VK; Nash. Kevin T KT; Hurst. Douglas R DR; Rama K...

The study shows that the kisspeptin‑54 peptide, which is linked to puberty and cancer‑spread suppression, doesn’t have a fixed shape in water or even in membrane‑like environments, but it still works biologically. Its flexible, mostly disordered structure might let it bind many different targets.

Utility 2
pubmed Aug 15, 2009

KiSS1 suppresses TNFalpha-induced breast cancer cell invasion via an inhibition of RhoA-mediated NF-kappaB activation.

Cho. Sung-Gook SG; Li. Dali D; Stafford. Lewis J LJ; Luo. Jian J; Rodriguez-Villanueva. Melissa M; W...

The study found that kisspeptin-10 (KP10) can block a specific inflammation signal (TNF‑alpha) that normally makes breast cancer cells more mobile and invasive. By doing this, KP10 reduces the activity of a protein chain (RhoA → NF‑kappaB) that drives cancer cell movement, but it doesn’t noticeably affect how fast the cancer cells grow.

Utility 2
pubmed 2010

Physiological roles of the kisspeptin/GPR54 system in the neuroendocrine control of reproduction.

Pineda. Rafael R; Aguilar. Enrique E; Pinilla. Leonor L; Tena-Sempere. Manuel M

Kisspeptin is a tiny protein that acts like a master switch for the hormones that control puberty, fertility and the whole reproductive system. It talks to a receptor called GPR54, which then tells the brain to release GnRH, the hormone that starts the cascade of reproductive hormones. The system also listens to the body’s energy status, so when you’re low on calories it can shut down fertility. This review just sums up what we know so far, without giving any new drug or dosage advice.

Utility 2
pubmed Aug 25, 2010

Kisspeptins: bridging energy homeostasis and reproduction.

Castellano. Juan M JM; Bentsen. Agnete H AH; Mikkelsen. Jens D JD; Tena-Sempere. Manuel M

Kisspeptin is a brain peptide that helps connect how much energy your body has with the hormones that control puberty and fertility. It appears to be a key link in how the fat‑signal hormone leptin talks to the reproductive system, and other metabolic signals like ghrelin and neuropeptide Y can also affect it.

Utility 2
pubmed Oct 23, 2008

Kisspeptin-10 facilitates a plasma membrane-driven calcium oscillator in gonadotropin-releasing hormone-1 neurons.

Constantin. Stephanie S; Caligioni. Claudia Simone CS; Stojilkovic. Stanko S; Wray. Susan S

Kisspeptin‑10 can kick‑start calcium waves in brain cells that control reproductive hormone release, doing so by turning on a membrane‑based oscillator that needs sodium channels and a specific signaling pathway. The work was done in mouse tissue, not humans, and shows how the peptide works at a cellular level rather than giving a ready‑to‑use protocol.

Utility 2
pubmed 2008

Peripheral administration of kisspeptin-10 increases plasma concentrations of GH as well as LH in prepubertal Holstein heifers.

Kadokawa. H H; Matsui. M M; Hayashi. K K; Matsunaga. N N; Kawashima. C C; Shimizu. T T; Kida. K K; M...

Injecting kisspeptin-10 into young dairy cows caused short‑term spikes in both growth hormone (GH) and luteinizing hormone (LH), showing the peptide can affect the body’s growth and reproductive systems, but the study was done in pre‑pubertal cattle, not humans.