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Kisspeptin-10

KP-10, Metastin (45-54), Kisspeptin-10 (human), KiSS-1

Kisspeptin-10 is a decapeptide that activates the KISS1R receptor to stimulate GnRH release, regulating the reproductive hormone axis and fertility.

Quick Stats
Studies 877
Trials 47
Formula C63H83N17O14
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Utility 2
pubmed Feb 24, 2014

Kisspeptin modulates fertilization capacity of mouse spermatozoa.

Hsu. Meng-Chieh MC; Wang. Jyun-Yuan JY; Lee. Yue-Jia YJ; Jong. De-Shien DS; Tsui. Kuan-Hao KH; Chiu....

In mice, the hormone kisspeptin and its receptor are found in sperm and egg‑related cells. Adding a short kisspeptin peptide (kisspeptin‑10) makes sperm calcium levels go up, which is important for fertilization, while blocking kisspeptin lowers IVF success. This points to kisspeptin playing a role in the fertilization process.

Utility 2
pubmed Jan 7, 2011

Control of GnRH secretion: one step back.

Clarke. Iain J IJ

This review explains that the brain’s GnRH hormone, which controls reproduction, is regulated by upstream neurons rather than directly by sex hormones. Kisspeptin neurons act as the main bridge for sex‑steroid feedback to GnRH, while GnIH neurons can suppress GnRH and also affect the pituitary. The paper highlights these pathways as key steps in how stress, nutrition, and seasons influence reproductive function.

Utility 2
pubmed Jun 9, 2011

Characterization of the kisspeptin system in human spermatozoa.

Pinto. F M FM; Cejudo-Román. A A; Ravina. C G CG; Fernández-Sánchez. M M; Martín...

Researchers found that the hormone kisspeptin and its receptor are actually present in human sperm cells. When sperm are exposed to kisspeptin in the lab, calcium levels rise slowly, and sperm movement changes in a two‑phase pattern – first it speeds up, then it slows down, and there’s a brief boost in a vigorous swimming style called hyperactivation. However, kisspein doesn’t trigger the sperm’s acrosome reaction, which is needed for fertilization, and blocking its receptor stops these effects.

Utility 2
pubmed Mar 31, 2011

Gene structure analysis of kisspeptin-2 (Kiss2) in the Senegalese sole (Solea senegalensis): characterization of two splice variants of Kiss2, and novel evidence for metabolic regulation of kisspeptin signaling in non-mammalian species.

Mechaly. Alejandro S AS; Viñas. Jordi J; Piferrer. Francesc F

This fish study found that the sole has two versions of the kisspeptin gene – one that works and one that doesn’t – and that when the fish fasts, the working version goes up in the brain and triggers higher reproductive hormone signals, linking food status to reproduction.

Utility 2
pubmed Jun 6, 2011

Transcriptional regulation of the human KiSS1 gene.

Mueller. Johanna K JK; Dietzel. Anja A; Lomniczi. Alejandro A; Loche. Alberto A; Tefs. Katrin K; Kie...

The paper maps how the kisspeptin gene (KiSS1) is turned on and off in brain cells that control puberty, showing which proteins boost its activity and which suppress it, but it doesn’t give any direct tips for using kisspeptin as a supplement or therapy.

Utility 2
pubmed May 29, 2013

In vivo recordings of GnRH neuron firing reveal heterogeneity and dependence upon GABAA receptor signaling.

Constantin. Stephanie S; Iremonger. Karl J KJ; Herbison. Allan E AE

In live mice, most GnRH cells that control fertility fire on their own, but they do so in many different ways. Giving kisspeptin (a short peptide) reliably turns these cells on, while drugs that change GABA‑A receptor activity can either boost or shut down their firing. This shows that the brain’s reproductive switch is highly variable and heavily dependent on GABA signaling.

Utility 2
pubmed Jul 18, 2014

A "kiss" before conception: triggering ovulation with kisspeptin-54 may improve IVF.

Young. Steven L SL

A 30‑year‑old woman with PCOS used kisspeptin‑54 to trigger ovulation for IVF and ended up with a severe form of ovarian hyperstimulation syndrome, including massive fluid buildup in her abdomen. The case shows that while kisspeptin can be used to induce ovulation, it can still cause dangerous side effects if the ovaries are overly stimulated.

Utility 2
pubmed Apr 1, 2012

Evaluation of serum kisspeptin levels in girls in the diagnosis of central precocious puberty and in the assessment of pubertal suppression.

Demirbilek. Huseyin H; Gonc. Elmas Nazli EN; Ozon. Alev A; Alikasifoglu. Ayfer A; Kandemir. Nurgun N

The study found that girls with early puberty have higher blood levels of the hormone kisspeptin, and those levels drop when treatment successfully stops puberty. This suggests kisspeptin could help doctors confirm early puberty and track if treatment is working, but it doesn’t give a new way to boost health or performance for most people.

Utility 2
pubmed Nov 8, 2010

Kisspeptin-evoked calcium signals in isolated primary rat gonadotropin- releasing hormone neurones.

Kroll. Heike H; Bolsover. Stephen S; Hsu. Judith J; Kim. Soo-Hyun SH; Bouloux. Pierre-Marc PM

The study shows that kisspeptin-10 makes certain brain cells that control reproductive hormones (GnRH neurons) take up more calcium. Most of this calcium comes in through channels that don’t need electrical spikes, while a smaller part comes from voltage‑gated channels that are triggered by sodium spikes.

Utility 2
pubmed Aug 22, 2012

Effects of kisspeptin-10 on lipid metabolism in cultured chicken hepatocytes.

Wu. J J; Fu. W W; Huang. Y Y; Ni. Y Y

In a lab study using chicken liver cells, the peptide kisspeptin‑10 (Kp‑10) at a concentration of 100 nM boosted the cells' production of triglycerides and cholesterol‑carrying particles without killing the cells. It also changed the activity of several genes that control fat metabolism, although the protein that drives fat synthesis (SREBP‑1) went up even though its gene level went down.

Utility 2
pubmed Nov 26, 2010

Intraperitoneal kisspeptin-10 administration induces dose-dependent degenerative changes in maturing rat testes.

Ramzan. Faiqah F; Qureshi. Irfan Zia IZ

A study in young male rats found that giving kisspeptin-10 repeatedly for two weeks lowered key hormones (LH and testosterone) and caused serious damage to the testes, including fewer sperm cells and structural degeneration. The harmful effects were seen at doses as low as 1 ng per injection, and got worse with higher doses.

Utility 2
pubmed Sep 18, 2012

Deciphering puberty: novel partners, novel mechanisms.

Tena-Sempere. Manuel M

This review explains that the kisspeptin system in the brain is a major driver of puberty and that its activity is influenced by the body’s energy balance and other neuropeptides, with epigenetic factors also playing a role. It doesn’t give any direct instructions for using kisspeptin-10, but it highlights how metabolism and hormones interact during development.

Utility 2
pubmed Aug 17, 2012

Low degree of overlap between kisspeptin, neurokinin B, and dynorphin immunoreactivities in the infundibular nucleus of young male human subjects challenges the KNDy neuron concept.

Hrabovszky. Erik E; Sipos. Máté T MT; Molnár. Csilla S CS; Ciofi. Philippe P; Borsay....

In young men, the brain cells that make kisspeptin, neurokinin B, and dynorphin are mostly separate, unlike what’s seen in animals. This means the popular “KNDy neuron” idea doesn’t fully apply to humans, so animal‑based tricks for tweaking hormone pulses may not work the same way in people.

Utility 2
pubmed Feb 24, 2012

Prognostic role of KiSS-1 and possibility of therapeutic modality of metastin, the final peptide of the KiSS-1 gene, in urothelial carcinoma.

Takeda. Toshikazu T; Kikuchi. Eiji E; Mikami. Shuji S; Suzuki. Eriko E; Matsumoto. Kazuhiro K; Miyaj...

The study shows that higher levels of the KiSS-1 gene are linked to better outcomes in a type of bladder cancer, and that giving the peptide metastin (related to kisspeptin‑10) to mice reduces tumor spread and improves survival, mainly by blocking a cell‑signaling pathway (NF‑κB) that helps cancer invade tissue.

Utility 2
pubmed Feb 16, 2012

Inactivating KISS1 mutation and hypogonadotropic hypogonadism.

Topaloglu. A Kemal AK; Tello. Javier A JA; Kotan. L Damla LD; Ozbek. Mehmet N MN; Yilmaz. M Bertan M...

A genetic mutation that disables the kisspeptin protein caused a family to fail puberty, proving that functional kisspeptin is essential for the hormone signals that start reproduction.

Utility 2
pubmed Jan 18, 2012

Kisspeptin-GPR54 signaling in mouse NO-synthesizing neurons participates in the hypothalamic control of ovulation.

Hanchate. Naresh Kumar NK; Parkash. Jyoti J; Bellefontaine. Nicole N; Mazur. Danièle D; Colledg...

The study shows that kisspeptin talks to brain cells that make nitric oxide (NO) to help trigger the hormone surge that leads to ovulation in mice. This interaction happens in a specific brain area and involves a signaling pathway (AKT) that activates the NO‑making enzyme. While the work is done in mice, it suggests that kisspeptin’s effect on fertility may depend on NO signaling.

Utility 2
pubmed Jan 27, 2011

Kisspeptin activates the hypothalamic-adenohypophyseal-gonadal axis in prepubertal ewe lambs.

Redmond. J S JS; Macedo. G G GG; Velez. I C IC; Caraty. A A; Williams. G L GL; Amstalden. M M

In young sheep, giving kisspeptin-10 through an IV caused quick bursts of the hormone LH, raised estrogen levels, and briefly triggered a luteal‑like phase, but it didn’t speed up the overall timing of puberty. The effect was short‑lived and the study was done in lambs, not people.

Utility 2
pubmed Aug 17, 2012

KISS1 expression in human female adipose tissue.

Cockwell. Heather H; Wilkinson. Diane A DA; Bouzayen. Renda R; Imran. Syed A SA; Brown. Russell R; W...

Researchers found that the gene for kisspeptin (KISS1) is active in women's fat tissue, especially under the skin, and that higher levels in belly fat are linked to higher BMI. This suggests that kisspeptin isn’t just a brain hormone but may also be made by fat cells.

Utility 2
pubmed 2011

Novel role of puberty onset protein kisspeptin as an anticoagulation peptide.

Qureshi. Irfan Zia IZ; Kanwal. Sobia S

Researchers found that kisspeptin-10, a peptide normally involved in puberty, can thin the blood in rats and also affects human blood samples in the lab, making it take longer to clot. The effect grows with higher doses and seems linked to lower calcium levels and fewer platelets, but the study is still early‑stage and only done in animals and test tubes.

Utility 2
pubmed Sep 15, 2010

Kisspeptin-10 inhibits bone-directed migration of GPR54-positive breast cancer cells: Evidence for a dose-window effect.

Olbrich. Teresa T; Ziegler. Elke E; Türk. Gregor G; Schubert. Antje A; Emons. Günter G; Gr...

Researchers found that a short peptide called kisspeptin‑10 can block breast cancer cells that have the GPR54 receptor from moving toward bone in lab dishes. The effect only shows up within a narrow concentration range (about one trillionth to one hundred‑billionth of a mole). It works by lowering the cancer cells' CXCR4 receptor and the bone‑cell signal (SDF‑1) that normally attracts them.