Menu
Peptide Database
Results
No peptides found
Featured

Use search to browse all 100+ peptides

Kisspeptin-10

KP-10, Metastin (45-54), Kisspeptin-10 (human), KiSS-1

Kisspeptin-10 is a decapeptide that activates the KISS1R receptor to stimulate GnRH release, regulating the reproductive hormone axis and fertility.

Quick Stats
Studies 877
Trials 47
Formula C63H83N17O14
Clear All
Utility 3
pubmed Jun 3, 2014

Reproduction Symposium: hypothalamic neuropeptides and the nutritional programming of puberty in heifers.

Amstalden. M M; Cardoso. R C RC; Alves. B R C BR; Williams. G L GL

The study shows that how much and what young cows eat changes brain signals (like kisspeptin, NPY, and α‑MSH) that control the start of puberty. Faster weight gain speeds up puberty, while restricted growth delays it. These brain pathways adapt structurally and genetically to nutrition, suggesting diet can program reproductive timing.

Utility 3
pubmed 2013

Effects of environmental endocrine disruptors and phytoestrogens on the kisspeptin system.

Patisaul. Heather B HB

The review shows that chemicals like BPA, PCBs and the plant estrogen genistein can mess up the kisspeptin system, which is a key hormone pathway for puberty, fertility and metabolism. These disruptions depend on the brain region, sex, and the specific chemical, and they can cause early puberty in girls, irregular cycles, and even affect mood and metabolism.

Utility 3
pubmed Jul 18, 2014

Kisspeptin-54 triggers egg maturation in women undergoing in vitro fertilization.

Jayasena. Channa N CN; Abbara. Ali A; Comninos. Alexander N AN; Nijher. Gurjinder M K GM; Christopou...

A single shot of kisspeptin‑54 can safely cause the hormone surge that matures eggs in women undergoing IVF, with more mature eggs seen at higher doses and about a quarter of treated women achieving pregnancy.

Utility 3
pubmed Apr 19, 2013

Exploring the pathophysiology of hypogonadism in men with type 2 diabetes: kisspeptin-10 stimulates serum testosterone and LH secretion in men with type 2 diabetes and mild biochemical hypogonadism.

George. Jyothis T JT; Veldhuis. Johannes D JD; Tena-Sempere. Manuel M; Millar. Robert P RP; Anderson...

In a tiny study, giving men with type‑2 diabetes and low testosterone a short burst of the hormone‑like peptide kisspeptin‑10 raised their luteinising hormone (LH) and, after a longer infusion, also lifted their testosterone levels. The effect was seen both in healthy volunteers and the diabetic participants, showing kisspeptin can kick‑start the body’s own testosterone production, but the work was done with IV doses and involved only a handful of people.

Utility 3
pubmed Aug 10, 2011

Evidence from the agonadal juvenile male rhesus monkey (Macaca mulatta) for the view that the action of neurokinin B to trigger gonadotropin-releasing hormone release is upstream from the kisspeptin receptor.

Ramaswamy. Suresh S; Seminara. Stephanie B SB; Plant. Tony M TM

In young male monkeys without testes, constantly giving kisspeptin-10 made the kisspeptin receptor stop working and also blocked the hormone‑releasing effect of a related peptide (NKB). Stopping the kisspeptin infusion let the system recover. Doing the opposite—continuously giving the NKB‑mimic—did not stop kisspeptin from triggering hormone release. This shows NKB works before kisspeptin in the chain that tells the brain to release reproductive hormones.

Utility 3
pubmed Sep 12, 2013

Twice-daily subcutaneous injection of kisspeptin-54 does not abolish menstrual cyclicity in healthy female volunteers.

Jayasena. C N CN; Comninos. A N AN; Nijher. G M K GM; Abbara. A A; De Silva. A A; Veldhuis. J D JD;...

A short, one‑week course of twice‑daily kisspeptin‑54 injections given during the middle of the menstrual cycle did not stop periods in healthy women. Instead, it made the overall cycle a little shorter and caused the hormone surge that triggers ovulation to happen a couple of days earlier.

Utility 3
pubmed Dec 23, 2011

GPR54 peptide agonists stimulate insulin secretion from murine, porcine and human islets.

Bowe. James E JE; Foot. Victoria L VL; Amiel. Stephanie A SA; Huang. Gao Cai GC; Lamb. Morgan W MW;...

The study found that short kisspeptin peptides (kisspeptin‑10 and kisspeptin‑13) quickly boost insulin release from isolated pancreas cells in mice, pigs, rats and humans when glucose is high. The effect is fast, reversible, and works across species, suggesting the peptides act directly on insulin‑producing cells. Earlier reports of inhibition may have been due to different lab methods.

Utility 3
pubmed Apr 2, 2012

Differential response of the primate HPG axis to N-methyl-D, L-aspartate, but not to Kisspeptin challenge under euglycemic and hypoglycemic conditions.

Wahab. F F; Zaman. W-uz WU; Shahab. M M

In male monkeys, giving the hormone‑boosting peptide kisspeptin‑10 raised testosterone just as well whether the animals had normal blood sugar or were made low on sugar by insulin. Other stimulants that rely on excitatory amino acids worked less well when blood sugar was low, but kisspeptin’s effect stayed strong.

Utility 3
pubmed Dec 6, 2010

Study on the effect of peripheral kisspeptin administration on basal and glucose-induced insulin secretion under fed and fasting conditions in the adult male rhesus monkey (Macaca mulatta).

Wahab. F F; Riaz. T T; Shahab. M M

Giving a short burst of kisspeptin‑10 (a hormone that normally helps control reproduction) to adult male rhesus monkeys didn’t change their normal insulin levels, but it made their pancreas release more insulin when glucose was given, whether the animals were fed or fasting. This hints that kisspeptin might boost the body’s insulin response to sugar.

Utility 3
pubmed Jun 13, 2011

Peripheral kisspeptin reverses short photoperiod-induced gonadal regression in Syrian hamsters by promoting GNRH release.

Ansel. L L; Bentsen. A H AH; Ancel. C C; Bolborea. M M; Klosen. P P; Mikkelsen. J D JD; Simonneaux....

Giving kisspeptin (a hormone that tells the brain to release reproductive signals) as a quick injection into the body can wake up the reproductive system in hamsters that have gone dormant because of short winter days, raising testosterone levels. However, a slow‑release method didn’t work, so timing and dosing matter. The findings hint that short, repeated doses might be needed if you ever try kisspeptin to boost hormones, but it’s still an animal study and not proven for people.

Utility 3
pubmed Sep 4, 2009

The mammalian target of rapamycin as novel central regulator of puberty onset via modulation of hypothalamic Kiss1 system.

Roa. J J; Garcia-Galiano. D D; Varela. L L; Sánchez-Garrido. M A MA; Pineda. R R; Castellano. J...

The study shows that the brain’s mTOR pathway helps start puberty by controlling the kisspeptin system. Turning mTOR on with the amino acid leucine boosts LH hormone release, while blocking mTOR with rapamycin delays puberty and lowers reproductive hormones in young female rats. Even when mTOR is blocked, the animals still respond to kisspeptin-10, meaning the basic GnRH system stays functional.

Utility 3
pubmed May 10, 2012

Kisspeptin administration to women: a window into endogenous kisspeptin secretion and GnRH responsiveness across the menstrual cycle.

Chan. Yee-Ming YM; Butler. James P JP; Sidhoum. Valerie F VF; Pinnell. Nancy E NE; Seminara. Stephan...

Giving kisspeptin to women triggers a quick rise in LH (the hormone that tells the ovaries to release eggs) but only when they are in the mid‑luteal or pre‑ovulatory part of their cycle. In the early follicular phase (right after the period starts) the response is weak and giving more kisspeptin doesn’t help. This means the body’s own kisspeptin levels are already high early in the cycle, so extra kisspeptin doesn’t add much.

Utility 3
pubmed Sep 27, 2012

Kisspeptins in human reproduction-future therapeutic potential.

Kaur. Kulvinder Kochar KK; Allahbadia. Gautam G; Singh. Mandeep M

Kisspeptin-10 is a hormone that helps control the brain's reproductive center. It plays a big role in starting puberty, regulating fertility, and linking metabolism to reproductive signals. Researchers think that drugs that mimic or block kisspeptin could someday treat delayed puberty, certain forms of infertility, hormone‑related amenorrhea, and maybe even help with some cancers or eating disorders, but real‑world dosing and safety are still being worked out.

Utility 3
pubmed Oct 10, 2008

Comparison of the effects of peripherally administered kisspeptins.

Mikkelsen. Jens D JD; Bentsen. Agnete H AH; Ansel. Laura L; Simonneaux. Valerie V; Juul. Anders A

In male mice, giving kisspeptin peptides (both short 10‑amino‑acid and longer versions) under the skin quickly raises blood testosterone, and the human versions work just as well as the mouse ones. Longer peptides act a bit slower but keep testosterone up longer, and the effect depends on the body’s GnRH system, not directly on the brain cells that make GnRH.

Utility 3
pubmed Oct 15, 2010

Neurobiological mechanisms underlying GnRH pulse generation by the hypothalamus.

Maeda. Kei-Ichiro K; Ohkura. Satoshi S; Uenoyama. Yoshihisa Y; Wakabayashi. Yoshihiro Y; Oka. Yoshit...

The paper explains that the brain releases the hormone GnRH in two ways – a big surge for ovulation and regular pulses that keep the reproductive system running. These pulses are fine‑tuned by hormones like estrogen and by things like light, food, and stress. The authors argue that a group of brain cells that make kisspeptin, especially in the arcuate nucleus, are the main drivers of these GnRH pulses.

Utility 3
pubmed Jan 16, 2010

Insights into the mechanism by which kisspeptin stimulates a preovulatory LH surge and ovulation in seasonally acyclic ewes: potential role of estradiol.

Sébert. M-E ME; Lomet. D D; Saïd. S Ben SB; Monget. P P; Briant. C C; Scaramuzzi. R J RJ;...

Giving sheep a steady IV dose of kisspeptin-10 for many hours caused a big rise in the hormone LH that leads to ovulation, but only when the treatment also raised estrogen levels. The longer the kisspeptin was infused, the more likely the animals were to have this LH surge.

Utility 3
pubmed Mar 4, 2008

Sex steroids and leptin regulate the "first Kiss" (KiSS 1/G-protein-coupled receptor 54 system) in human gonadotropin-releasing-hormone-secreting neuroblasts.

Morelli. Annamaria A; Marini. Mirca M; Mancina. Rosa R; Luconi. Michaela M; Vignozzi. Linda L; Fibbi...

The study shows that kisspeptin can make GnRH‑releasing cells fire more hormone, while estrogen dampens, and androgens and leptin boost the kisspeptin system. In simple terms, sex hormones and the fat‑derived hormone leptin work together to turn on a key pathway that starts puberty, but the work was done in fetal brain cells, not in living adults.

Utility 3
pubmed Jul 4, 2008

Kisspeptins and the control of gonadotropin secretion in humans.

Jayasena. C N CN; Dhillo. W S WS; Bloom. S R SR

Kisspeptin is a naturally occurring peptide that, when given to healthy people, quickly raises the hormones that tell the testes and ovaries to produce sex hormones, without obvious side effects. This shows it could be a safe way to tweak the reproductive hormone system, which influences things like muscle growth, mood, and metabolism, but the study doesn’t give a clear dosing plan for DIY use.

Utility 3
pubmed 2007

Leptin in reproduction.

Blüher. Susann S; Mantzoros. Christos S CS

Leptin, a hormone that tells the brain about energy stores, also helps start puberty and keep the reproductive system working. New animal and early human studies suggest that leptin works through kisspeptin‑producing neurons (KiSS1) to control fertility, and that giving leptin can fix reproductive problems caused by low leptin levels.