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Kisspeptin-10

KP-10, Metastin (45-54), Kisspeptin-10 (human), KiSS-1

Kisspeptin-10 is a decapeptide that activates the KISS1R receptor to stimulate GnRH release, regulating the reproductive hormone axis and fertility.

Quick Stats
Studies 877
Trials 47
Formula C63H83N17O14
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Utility 2
pubmed Nov 23, 2020

Kisspeptin-54 Accurately Identifies Hypothalamic Gonadotropin-Releasing Hormone Neuronal Dysfunction in Men with Congenital Hypogonadotropic Hypogonadism.

Abbara. Ali A; Eng. Pei Chia PC; Phylactou. Maria M; Clarke. Sophie A SA; Mills. Edouard E; Chia. Ge...

The study shows that a single IV dose of kisspeptin‑54 triggers a strong rise in luteinizing hormone (LH) in healthy men, but almost no response in men with a genetic form of low hormone production, making it a precise test for hypothalamic function.

Utility 2
pubmed Oct 29, 2020

Associations of serum kisspeptin levels with metabolic and reproductive parameters in men.

Sitticharoon. Chantacha C; Mutirangura. Pornthira P; Chinachoti. Thitima T; Iamaroon. Arissara A; Tr...

The study found that men with higher body weight and obesity have higher levels of kisspeptin in their blood, and these levels go up together with insulin, insulin resistance, and leptin, while they go down with a hormone called LH. No kisspeptin was detected in the spinal fluid. This suggests kisspein might play a role in how the body handles metabolism, especially in overweight people.

Utility 2
pubmed Dec 17, 2019

The Roles of the Amygdala Kisspeptin System.

Mills. Edouard G A EGA; O'Byrne. Kevin T KT; Comninos. Alexander N AN

This review explains that kisspeptin, a hormone best known for controlling reproduction, is also found in the amygdala—a brain area linked to emotions and behavior. In the amygdala, kisspeptin helps set the timing of puberty, shapes the pattern of reproductive hormone release, and ties those hormones to sexual and social behaviors. The authors suggest that targeting this brain system could lead to new treatments for reproductive or psychosexual problems, but they don’t give any specific dosing or DIY advice.

Utility 2
pubmed Dec 17, 2019

Role of Kisspeptin and NKB in Puberty in Nonhuman Primates: Sex Differences.

Garcia. James P JP; Keen. Kim L KL; Seminara. Stephanie B SB; Terasawa. Ei E

In monkey brains, the peptide kisspeptin-10 (and a related molecule called NKB) can boost the release of the hormone GnRH, which controls reproductive hormones. Girls' brains respond more strongly to kisspeptin than boys', and during puberty the wiring between kisspeptin and NKB changes – females develop a two‑way communication loop, while males rely mainly on kisspeptin alone. Both signals help increase GnRH during puberty, but they don’t start puberty on their own.

Utility 2
pubmed Nov 15, 2019

Intraperitoneal Treatment of Kisspeptin Suppresses Appetite and Energy Expenditure and Alters Gastrointestinal Hormones in Mice.

Dong. Tien S TS; Vu. John P JP; Oh. Suwan S; Sanford. Daniel D; Pisegna. Joseph R JR; Germano. Patri...

In mice, a single injection of the peptide kisspeptin-10 lowered how much they ate, made them eat fewer and smaller meals, and reduced their overall energy use. At the same time, it raised blood levels of insulin, leptin, resistin and good cholesterol (HDL) and made their bodies burn more carbs than fat. The study suggests kisspeptin can influence appetite and metabolism, but it was done by injecting the peptide directly into the abdomen of mice, which isn’t a typical way people could use it.

Utility 2
pubmed Mar 7, 2020

Roles of the kisspeptin/GPR54 system in pathomechanisms of atherosclerosis.

Watanabe. Takuya T; Sato. Kengo K

Kisspeptin-10 (KP-10) and its receptor GPR54 are found in high amounts in artery plaques and seem to make those plaques grow faster and become more unstable, which could lead to heart attacks. In lab cells, KP-10 blocks healthy blood‑vessel cell growth, pushes immune cells to stick to vessels, and makes fat‑laden foam cells that are a hallmark of atherosclerosis. In mice that are prone to artery disease, giving KP-10 speeds up plaque formation, but blocking GPR54 with a drug called P234 stops those bad effects.

Utility 2
pubmed Jun 8, 2020

Relevance of <i>KISS1</i> gene polymorphisms in susceptibility to polycystic ovary syndrome and its associated endocrine and metabolic disturbances.

Daghestani. M H MH; Daghestani. M H MH; Daghistani. M M; Ambreen. K K; Almuammar. M N MN; Al Neghery...

A study found a specific genetic change in the KISS1 gene (rs1213704663C>G) that’s linked to a higher chance of polycystic ovary syndrome (PCOS) and to higher LH and estrogen levels, but it doesn’t change kisspeptin levels. This isn’t a treatment, just a genetic risk marker.

Utility 2
pubmed Jul 8, 2021

Effect of anti-M&#xfc;llerian hormone in hypothalamic Kiss-1- and GnRH-producing cell models.

Oride. Aki A; Kanasaki. Haruhiko H; Tumurbaatar. Tuvshintugs T; Tumurgan. Zolzaya Z; Okada. Hiroe H;...

The study shows that adding anti‑Müllerian hormone (AMH) to hypothalamic cells boosts the production of GnRH (the hormone that tells the pituitary to release reproductive hormones) but does not change the amount of kisspeptin (Kiss‑1) made by those cells. In fact, AMH can block the increase in Kiss‑1 that normally happens when you add kisspeptin‑10. This suggests AMH can influence the reproductive hormone cascade by promoting GnRH while dampening kisspeptin‑driven signals.

Utility 2
pubmed Jul 24, 2020

The content of gonadotropin-releasing hormone (GnRH), kisspeptin, and estrogen receptors (ER&#x3b1;/ER&#x3b2;) in the anteromedial hypothalamus displays daily variations throughout the rat estrous cycle.

Olvera-Ju&#xe1;rez. Esteban E; Silva. Carlos-Camilo CC; Flores. Ang&#xe9;lica A; Arrieta-Cruz. Isabe...

In rats, the amount of kisspeptin and related hormones in a specific brain region changes throughout the day and across the reproductive cycle, and the right side of that region usually has higher levels. This shows that hormone levels are not constant but follow daily and cycle‑related patterns.

Utility 2
pubmed Apr 6, 2020

Hypothalamic and brain stem neurochemical profile in anorectic rats after peripheral administration of kisspeptin-10 using <sup>1</sup> H-nmr spectroscopy in vivo.

Skowron. Kamil K; Jasi&#x144;ski. Krzysztof K; Kurnik-&#x141;ucka. Magdalena M; Stach. Paulina P; Ka...

In a rat model of anorexia, giving the peptide kisspeptin-10 under the skin helped the animals eat more and changed several brain chemicals linked to energy use. The study shows kisspeptin can affect appetite by tweaking signals in the hypothalamus, but it’s only been tested in mice, not people.

Utility 2
pubmed May 20, 2024

[Notch1/Akt/Foxo1 Pathway Regulated by Kisspeptin Is Involved in Endometrial Decidualization in Patients With Recurrent Spontaneous Abortion].

Yang. Yanhong Y; Zhang. Jianliang J; Li. Dongxiao D; Liu. Cuiping C; Guo. Rong R; Xiao. Yi Y; Zhou....

The study shows that women who have had repeated miscarriages have lower levels of the hormone‑like peptide kisspeptin. Adding a short form of kisspeptin (kisspeptin‑10) to uterine cells in the lab makes them change into a state that supports pregnancy, and giving kisspeptin‑10 to mice that normally lose embryos reduces those losses. The effect works through a chain of cell‑signaling proteins called Notch1, Akt and Foxo1.

Utility 2
pubmed Jun 14, 2021

Safety Evaluation of KP-10 (Metastin 45-54) Following once Daily Intravenous Administration for 14 Days in Dog.

Terse. Pramod S PS; Peggins. James J; Seminara. Stephanie B SB

A study gave dogs a peptide called kisspeptin-10 (KP-10) once a day for two weeks and found no signs of toxicity even at the highest dose tested. The peptide cleared from the blood quickly, and the hormone LH spiked right after each dose but dropped over time. The dogs stayed in a non‑reproductive state throughout the experiment, and everything returned to normal after a two‑week recovery period.

Utility 2
pubmed Dec 12, 2021

Dose-Dependent Degeneration of Leydig Cells Following Kisspeptin-10 Administration: An Ultrastructural Study.

Ramzan. Faiqah F; Qureshi. Irfan Zia IZ; Ramzan. Muhammad Haris MH

In young male rats, giving kisspeptin-10 repeatedly lowered blood testosterone and caused damage to the testicular Leydig cells that make the hormone. The harmful effects got worse with higher doses. This suggests that chronic, high‑dose kisspeptin-10 could suppress testosterone production, at least in this animal model.

Utility 2
pubmed May 12, 2020

Chronic exposure to low dose of bisphenol A causes follicular atresia by inhibiting kisspeptin neurons in anteroventral periventricular nucleus in female mice.

Tang. Chuanfeng C; Zhang. Jia J; Liu. Peiyu P; Zhou. Yu Y; Hu. Qiaoyun Q; Zhong. Ying Y; Wang. Xiaol...

A study in female mice showed that long‑term low‑dose exposure to the plastic chemical BPA messes up the brain signals (kisspeptin neurons) that control the menstrual cycle, leading to fewer mature eggs and a longer low‑fertility phase. Giving the mice a small dose of the peptide kisspeptin‑10 straight into the brain fixed the hormone drops and restored the normal LH surge, suggesting kisspeptin can counteract BPA’s harmful effect on fertility in mice.

Utility 2
pubmed 2020

Kissorphin improves spatial memory and cognitive flexibility impairment induced by ethanol treatment in the Barnes maze task in rats.

Gibula-Tarlowska. Ewa E; Kotlinska. Jolanta H JH

In rats, a new peptide called kissorphin (based on kisspeptin-10) helped protect against memory problems caused by alcohol exposure and withdrawal. The biggest benefit was seen at the highest dose tested (10 nmol). The study suggests that tweaking the brain's opioid system might reverse alcohol‑related learning deficits, but it’s all animal work and not yet ready for human use.

Utility 2
pubmed Feb 17, 2021

KP-10/Gpr54 attenuates rheumatic arthritis through inactivating NF-&#x3ba;B and MAPK signaling in macrophages.

Wang. Dongsheng D; Wu. Zhixiang Z; Zhao. Chenglong C; Yang. Xinghai X; Wei. Haifeng H; Liu. Mingyao...

Researchers found that the short peptide kisspeptin‑10 (KP‑10) can calm down inflammation in immune cells and reduce arthritis symptoms in mice by blocking key inflammatory pathways. While the work shows promise, it’s still early‑stage lab work and not ready for personal use.

Utility 2
pubmed Jul 15, 2021

Mutual Interactions Between GnRH and Kisspeptin in GnRH- and Kiss-1-Expressing Immortalized Hypothalamic Cell Models.

Kanasaki. Haruhiko H; Tumurbaatar. Tuvshintugs T; Tumurgan. Zolzaya Z; Oride. Aki A; Okada. Hiroe H;...

The study shows that the short peptide kisspeptin‑10 can boost its own production and, in some hypothalamic cells, also increase the production of GnRH, another hormone that controls reproduction. This effect was seen in mouse brain cell lines and in rat fetal brain cells, suggesting a feedback loop between kisspeptin and GnRH in the brain.

Utility 2
pubmed Dec 28, 2021

The roles of kisspeptin and neurokinin B in GnRH pulse generation in humans, and their potential clinical application.

Anderson. Richard A RA; Millar. Robert P RP

The study shows that giving people a steady, high‑dose infusion of kisspeptin‑10 for about a day makes the brain release more frequent LH pulses (the hormone that tells the gonads to make sex hormones). This works in both men and women, even those with hormone problems, and the response doesn’t wear off after many hours.