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Kisspeptin-10

KP-10, Metastin (45-54), Kisspeptin-10 (human), KiSS-1

Kisspeptin-10 is a decapeptide that activates the KISS1R receptor to stimulate GnRH release, regulating the reproductive hormone axis and fertility.

Quick Stats
Studies 877
Trials 47
Formula C63H83N17O14
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Utility 2
pubmed Jun 18, 2019

The influence of a new derivate of kisspeptin-10 - Kissorphin (KSO) on the rewarding effects of morphine in the conditioned place preference (CPP) test in male rats.

Gibula-Tarlowska. E E; Kedzierska. E E; Piechura. K K; Silberring. J J; Kotlinska. J H JH

A new peptide called Kissorphin (KSO), made from kisspeptin‑10, was tested in rats and found to block the rewarding effects of morphine, a powerful opioid. It stopped rats from learning to like morphine, reduced the already‑learned preference, and prevented a relapse‑like response, without causing any preference or aversion on its own. The effect works through specific brain receptors (NPFF), and can be blocked by an antagonist, showing the mechanism is real, but the study was only in animals.

Utility 2
pubmed Oct 28, 2020

Impact of serum and follicular fluid kisspeptin and estradiol on oocyte maturity and endometrial thickness among unexplained infertile females during ICSI.

Rehman. Rehana R; Zafar. Amara A; Ali. Arzina Aziz AA; Baig. Mukhtiar M; Alam. Faiza F

The study found that higher levels of the hormone kisspeptin in both blood and the fluid around eggs (follicular fluid) during IVF cycles were linked to more mature eggs, thicker uterine lining, and better chances of pregnancy in women with unexplained infertility.

Utility 2
pubmed Jun 1, 2020

Kisspeptin and neurokinin B interactions in modulating gonadotropin secretion in women with polycystic ovary syndrome.

Skorupskaite. Karolina K; George. Jyothis T JT; Veldhuis. Johannes D JD; Millar. Robert P RP; Anders...

In women with PCOS, a 7‑day course of a neurokinin‑3 receptor blocker lowered baseline LH and FSH levels, but an infusion of kisspeptin‑10 still caused a strong rise in LH. The LH boost from kisspeptin was linked to estrogen levels unless the blocker was present, showing that kisspeptin can drive reproductive hormone release even when the NKB pathway is inhibited.

Utility 2
pubmed Sep 11, 2020

Kisspeptin preserves mitochondrial function by inducing mitophagy and autophagy in aging rat brain hippocampus and human neuronal cell line.

Mattam. Ushodaya U; Talari. Noble Kumar NK; Paripati. Arun Kumar AK; Krishnamoorthy. Thanuja T; Sepu...

The study shows that the brain peptide kisspeptin‑10 can boost the cleaning and recycling of mitochondria in brain cells, leading to more mitochondria, better energy production, and possibly improved memory in aging rats and human neuron cells. However, the work is still early‑stage and done in cells and animals, with no human dosing or safety data.

Utility 2
pubmed Dec 17, 2019

The Role of Kisspeptin in Sexual Behavior.

Hellier. Vincent V; Brock. Olivier O; Bakker. Julie J

In female mice, the hormone-like peptide kisspeptin is needed for normal sexual interest and the lordosis posture that signals readiness to mate. Removing kisspeptin stops these behaviors, but giving a single kisspeptin injection restores them. The peptide works through the usual GnRH pathway for preference, but a separate nitric‑oxide signal seems to drive the actual lordosis response.

Utility 2
pubmed May 19, 2020

Metabolic regulation of kisspeptin - the link between energy balance and reproduction.

Navarro. Víctor M VM

The review explains that the brain cells that make kisspeptin, a hormone that triggers reproductive signals, are tightly controlled by the body's energy status. When you have enough fuel (calories, fat stores), kisspeptin production goes up, helping fertility; when energy is low, production drops. The article also notes that kisspeptin can feed back to affect how the brain regulates appetite and metabolism, creating a two‑way link between metabolism and reproduction.

Utility 2
pubmed Apr 16, 2020

Characterization of Kisspeptin Neurons in the Human Rostral Hypothalamus.

Rumpler. Éva É; Skrapits. Katalin K; Takács. Szabolcs S; Göcz. Balázs B; Tr...

Researchers mapped kisspeptin‑producing neurons in the front part of the human hypothalamus and found they are influenced by estrogen, similar to what’s seen in animals. Men and young women have about the same number of these cells, but the count drops after menopause. These human cells are also chemically different from the ones studied in rodents.

Utility 2
pubmed May 11, 2021

Kisspeptin-54 attenuates oxidative stress and neuronal apoptosis in early brain injury after subarachnoid hemorrhage in rats via GPR54/ARRB2/AKT/GSK3β signaling pathway.

Huang. Yi Y; Guo. Yong Y; Huang. Lei L; Fang. Yuanjian Y; Li. Dujuan D; Liu. Rui R; Lu. Qin Q; Ren....

In rats that had a brain bleed, giving a form of the peptide kisspeptin-54 through the nose reduced brain damage, oxidative stress, and cell death, and helped the animals recover better over weeks. The protective effect depended on a specific receptor (GPR54) and downstream signaling proteins.

Utility 2
pubmed Dec 27, 2018

Age-dependent changes in the reproductive axis responsiveness to kisspeptin-10 administration in healthy men.

Ullah. Hamid H; Nabi. Ghulam G; Zubair. Hira H; Ullah. Rahim R; Shahab. Muhammad M

Giving a single IV dose of kisspeptin-10 (1 µg per kg body weight) makes the brain release more LH hormone in men of all ages, but only younger adult men see a rise in testosterone. As men get older, their testes become less responsive to the LH boost, so testosterone doesn't go up.

Utility 2
pubmed Dec 17, 2019

Does the KNDy Model for the Control of Gonadotropin-Releasing Hormone Pulses Apply to Monkeys and Humans?

Lehman. Michael N MN; He. Wen W; Coolen. Lique M LM; Levine. Jon E JE; Goodman. Robert L RL

Scientists think a group of brain cells that release kisspeptin, neurokinin B, and dynorphin (called KNDy neurons) helps control the timing of reproductive hormone bursts. This idea is well‑studied in rodents and some farm animals, but we still don’t know exactly how it works in monkeys or people. New drugs that target these KNDy signals are being tested for fertility and other hormone problems, so understanding this system in humans could become important.

Utility 2
pubmed Aug 23, 2021

Kisspeptin signaling and nNOS neurons in the VMHvl modulate lordosis behavior but not mate preference in female mice.

Bentefour. Yassine Y; Bakker. Julie J

In female mice, giving kisspeptin-10 directly into a specific brain area (the ventrolateral ventromedial hypothalamus) makes them more receptive to mating, and this effect seems to rely on neurons that produce nitric oxide. The same treatment does not change which male they prefer, and giving the hormone into other brain spots or giving GnRH does nothing.

Utility 2
pubmed 2020

Role of Kisspeptin in Regulation of Reproductive and Immune Reactions.

Gorbunova. O L OL; Shirshev. S V SV

Kisspeptin is a brain hormone that tells the body when to start puberty, release reproductive hormones, and adjust the immune system during pregnancy. It also appears to affect heart function in pregnant women and helps the immune system tolerate the fetus.

Utility 2
pubmed Jan 9, 2020

Kisspeptin Influence on Polycystic Ovary Syndrome-a Mini Review.

Araújo. Bruna Silva BS; Baracat. Maria Cândida P MCP; Dos Santos Simões. Ricardo R; d...

A short review found that women with polycystic ovary syndrome (PCOS) usually have higher blood levels of the peptide kisspeptin, and this is true regardless of whether they are lean or overweight.

Utility 2
pubmed Sep 21, 2017

Is there a role for kisspeptin in pathogenesis of polycystic ovary syndrome?

Gorkem. Umit U; Togrul. Cihan C; Arslan. Emine E; Sargin Oruc. Ayla A; Buyukkayaci Duman. Nuriye N

The study found that women with PCOS have higher blood levels of the peptide kisspeptin, and those levels go up when testosterone and DHEAS are high and down when FSH is high. This suggests kisspeptin is linked to the hormonal imbalances seen in PCOS, but the research doesn’t test any treatments or give dosing advice.

Utility 2
pubmed Aug 1, 2017

Metabonomics Approach to Assessing the Modulatory Effects of Kisspeptin-10 on Liver Injury Induced by Heat Stress in Rats.

Hou. Yuanlong Y; Wang. Xiaoyan X; Ping. Jihui J; Lei. Zhihai Z; Gao. Yingdong Y; Ma. Zhiyu Z; Jia. C...

In rats, giving kisspeptin-10 before a hot‑stress event helped protect the liver. The peptide reduced damage by boosting antioxidant defenses and normalising metabolism of purines and fats. The study shows a possible anti‑oxidant role for kisspeptin, but it’s an early animal experiment.

Utility 2
pubmed Jan 31, 2022

Lactational Amenorrhea: Neuroendocrine Pathways Controlling Fertility and Bone Turnover.

Calik-Ksepka. Anna A; Stradczuk. Monika M; Czarnecka. Karolina K; Grymowicz. Monika M; Smolarczyk. R...

During breastfeeding, high prolactin levels shut down kisspeptin neurons in the brain, which stops the normal GnRH and LH hormone pulses needed for ovulation, causing temporary infertility (lactational amenorrhea). This also leads to increased bone turnover to supply calcium to the baby, but bone density usually recovers after weaning. The lactational amenorrhea method (LAM) can be a reliable, low‑cost birth control if strict breastfeeding patterns are followed, but it’s not the same as just nursing.

Utility 2
pubmed Sep 1, 2017

A second dose of kisspeptin-54 improves oocyte maturation in women at high risk of ovarian hyperstimulation syndrome: a Phase 2 randomized controlled trial.

Abbara. Ali A; Clarke. Sophie S; Islam. Rumana R; Prague. Julia K JK; Comninos. Alexander N AN; Nara...

Giving a second injection of kisspeptin‑54 about 10 hours after the first one boosts the hormone surge that matures eggs, leading more women at high risk of ovarian hyperstimulation syndrome to get a good number of mature eggs, and it doesn’t raise the chance of severe side effects.

Utility 2
pubmed Jul 17, 2017

Cross-Linking Furan-Modified Kisspeptin-10 to the KISS Receptor.

Vannecke. Willem W; Ampe. Christophe C; Van Troys. Marleen M; Beltramo. Massimiliano M; Madder. Anne...

Scientists showed that a specially tweaked version of the kisspeptin-10 peptide can stick itself to its natural receptor on cell surfaces without using harmful UV light. The reaction happens inside living cells thanks to natural reactive oxygen species, making the process safe and efficient.

Utility 2
pubmed May 30, 2018

rs4889 polymorphism in KISS1 gene, its effect on polycystic ovary syndrome development and anthropometric and hormonal parameters in Saudi women.

Albalawi. Fadwa S FS; Daghestani. Maha H MH; Daghestani. Mazin H MH; Eldali. Abdelmoneim A; Warsy. A...

The study looked at a gene called KISS1 and a tiny protein called kisspeptin in Saudi women with polycystic ovary syndrome (PCOS). It found that women with PCOS had higher LH hormone levels and body weight, and a specific genetic variant (GG at rs4889) was more common in them and linked to higher kisspeptin and FSH levels. However, overall kisspeptin levels weren’t different from healthy women, and the research is small and observational, so it doesn’t give clear guidance on using kisspeptin for health improvement.