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Kisspeptin-10

KP-10, Metastin (45-54), Kisspeptin-10 (human), KiSS-1

Kisspeptin-10 is a decapeptide that activates the KISS1R receptor to stimulate GnRH release, regulating the reproductive hormone axis and fertility.

Quick Stats
Studies 877
Trials 47
Formula C63H83N17O14
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Utility 1
pubmed Aug 11, 2009

Kisspeptin-10, a KISS1-derived decapeptide, inhibits tumor angiogenesis by suppressing Sp1-mediated VEGF expression and FAK/Rho GTPase activation.

Cho. Sung-Gook SG; Yi. Zhengfang Z; Pang. Xiufeng X; Yi. Tingfang T; Wang. Ying Y; Luo. Jian J; Wu....

Kisspeptin‑10, a tiny protein fragment, was shown in lab experiments to stop new blood‑vessel growth that tumors need, shrinking tumor size in mice, but the work is all in cells and animals and doesn’t give any human dosing or safety info, so it isn’t ready for personal use.

Utility 1
pubmed Jun 20, 2011

Serum kisspeptin levels in Korean girls with central precocious puberty.

Rhie. Young Jun YJ; Lee. Kee Hyoung KH; Eun. So Hee SH; Choi. Byung Min BM; Chae. Hyun Wook HW; Kwon...

Researchers measured kisspeptin levels in Korean girls with early-onset puberty and found they were about twice as high as in normal pre‑pubertal girls. Higher kisspeptin was linked to stronger hormone responses that trigger puberty, suggesting it could be a useful blood marker for spotting early puberty.

Utility 1
pubmed Sep 8, 2011

Effects of kisspeptin-10 on progesterone secretion in cultured chicken ovarian granulosa cells from preovulatory (F1-F3) follicles.

Xiao. Yunqi Y; Ni. Yingdong Y; Huang. Yanbing Y; Wu. Jing J; Grossmann. Roland R; Zhao. Ruqian R

Scientists tested kisspeptin‑10 on chicken ovarian cells and found that a 100 nM dose raised progesterone output and cell health for up to two days, but after three days the hormone level fell. The peptide also turned on the genes that make steroid hormones, though the actual protein amounts didn’t change.

Utility 1
pubmed Apr 23, 2009

In vivo and in vitro structure-activity relationships and structural conformation of Kisspeptin-10-related peptides.

Gutiérrez-Pascual. Ester E; Leprince. Jérôme J; Martínez-Fuentes. Antonio J AJ;...

Scientists swapped out specific building blocks in the kisspeptin‑10 peptide and found that changes at two spots (positions 6 and 10) make the peptide far less able to trigger hormone release, showing those spots are essential for its activity.

Utility 1
pubmed Dec 21, 2009

Central administration of kisspeptin-10 inhibits natriuresis and diuresis induced by blood volume expansion in anesthetized male rats.

Han. Xu X; Yan. Ming M; An. Xiao-fei XF; He. Ming M; Yu. Jiang-yi JY

In a rat study, giving kisspeptin-10 directly into the brain stopped the usual increase in urine and salt loss that happens when blood volume is suddenly raised. This was linked to higher levels of the hormone vasopressin, but not to changes in another hormone (ANP) or kidney nerve signals. The findings are interesting for science but don’t give a clear way for people to use kisspeptin for fluid balance in everyday life.

Utility 1
pubmed Sep 21, 2009

Kisspeptin signaling in the brain.

Oakley. Amy E AE; Clifton. Donald K DK; Steiner. Robert A RA

Kisspeptin is a brain chemical that tells the reproductive system when to release hormones, affecting puberty, fertility, and hormone cycles. It works by activating GnRH neurons and is influenced by estrogen and testosterone. While it has roles beyond reproduction, the paper doesn’t give any direct ways to use it for health hacks or performance gains.

Utility 1
pubmed Aug 1, 2010

beta-Sheet aggregation of kisspeptin-10 is stimulated by heparin but inhibited by amphiphiles.

Nielsen. Søren B SB; Franzmann. Magnus M; Basaiawmoit. Rajiv V RV; Wimmer. Reinhard R; Mikkelse...

The study shows that the short hormone kisspeptin‑10 can clump together into amyloid‑like fibers when heparin is present, but these clumps are stopped by common surfactants. This behavior is a basic science finding and doesn’t give clear guidance on how to use kisspeptin for health or performance.

Utility 1
pubmed Oct 14, 2009

Molecular characterization and estrogen regulation of hypothalamic KISS1 gene in the pig.

Tomikawa. Junko J; Homma. Tamami T; Tajima. Shigeyuki S; Shibata. Takako T; Inamoto. Yoko Y; Takase....

Scientists mapped the kisspeptin gene in pig brains and saw how estrogen changes its activity. They found the active part of the peptide (kisspeptin‑10) is the same as in other animals, and estrogen boosts kisspeptin cells in one brain area while lowering them in another. This helps explain how estrogen controls reproductive hormones in pigs, but it doesn’t give direct tips for health hacks or dosing.

Utility 1
pubmed Jun 13, 2012

KiSS1 and its G-protein-coupled receptor GPR54 in cancer development and metastasis.

Cho. Sung-Gook SG; Li. Dali D; Tan. Kunrong K; Siwko. Stefan K SK; Liu. Mingyao M

The paper talks about a protein called kisspeptin (KiSS1) and its receptor GPR54, which are known for roles in reproduction but also show mixed effects on cancer spread. While early work suggested they might stop cancer cells from moving, newer research shows they can act in different ways, and their exact impact on cancer is still unclear.

Utility 1
pubmed Jul 21, 2009

Studies of the localisation of kisspeptin within the pituitary of the rhesus monkey (Macaca mulatta) and the effect of kisspeptin on the release of non-gonadotropic pituitary hormones.

Ramaswamy. S S; Gibbs. R B RB; Plant. T M TM

The study looked at where kisspeptin is found in the monkey pituitary and whether giving kisspeptin changes hormones like growth hormone, prolactin, thyroid‑stimulating hormone or cortisol. It found kisspeptin in some pituitary cells but, when injected, it did not alter the levels of those non‑reproductive hormones.

Utility 1
pubmed Sep 5, 2012

Plasma Kisspeptin-54 levels in gastric cancer patients.

Ergen. Arzu A; Canbay. Emel E; Bugra. Dursun D; Zeybek. Umit U; Yamaner. Sumer S; Bulut. Turker T

Researchers measured a hormone-like peptide called kisspeptin-54 in the blood of people with stomach cancer and found it was higher than in healthy people. While this could help doctors detect the disease, it doesn't give any direct advice on how to use kisspeptin-54 for improving health or performance.

Utility 1
pubmed Mar 25, 2009

Discovery of potent kisspeptin antagonists delineate physiological mechanisms of gonadotropin regulation.

Roseweir. Antonia K AK; Kauffman. Alexander S AS; Smith. Jeremy T JT; Guerriero. Kathryn A KA; Morga...

Scientists made molecules that block kisspeptin, a hormone that tells the brain to release reproductive hormones. In mice and monkeys these blockers stopped the brain signals that trigger puberty and reduced hormone spikes in several animal models. The work suggests these blockers could someday be used to treat conditions like early puberty, endometriosis, or hormone‑driven prostate cancer, but they aren’t a ready‑to‑use supplement or protocol for everyday health optimization.

Utility 1
pubmed Mar 20, 2009

Structural and functional multiplicity of the kisspeptin/GPR54 system in goldfish (Carassius auratus).

Li. Shuisheng S; Zhang. Yong Y; Liu. Yun Y; Huang. Xigui X; Huang. Weiren W; Lu. Danqi D; Zhu. Pei P...

Researchers studied two kisspeptin peptides in goldfish and found that one of them (gfKiss1-10) can raise a reproductive hormone (LH) when injected into mature females, but it doesn’t work directly on the pituitary cells. The other peptide (gfKiss2-10) was much weaker and showed no clear effect. These findings are specific to fish and don’t give clear guidance for human use.

Utility 1
pubmed Dec 16, 2009

Kisspeptin signalling in the hypothalamic arcuate nucleus regulates GnRH pulse generator frequency in the rat.

Li. Xiao-Feng XF; Kinsey-Jones. James S JS; Cheng. Yewsong Y; Knox. Alice M I AM; Lin. Yuanshao Y; P...

In rats, the peptide kisspeptin‑10 acting in a specific brain area (the arcuate nucleus) can boost the release of the hormone LH, which drives reproductive hormone cycles. Blocking kisspeptin there reduces LH pulses. This shows that kisspeptin signaling in that brain region is a key part of the natural rhythm that controls fertility hormones.

Utility 1
pubmed May 5, 2011

Functional interrelationship between the WASF3 and KISS1 metastasis-associated genes in breast cancer cells.

Teng. Yong Y; Liu. Mingyao M; Cowell. John K JK

In breast cancer cells, turning off the gene WASF3 makes the cells produce more of the KISS1 protein, which acts like a brake on cancer spread. This increase in KISS1 lowers the cells' ability to invade tissue and reduces activity of enzymes (MMP‑9) that help tumors break down surrounding material. The effect works by dampening a signaling pathway (NF‑κB) that normally promotes invasion.

Utility 1
pubmed Dec 1, 2009

Critical roles of kisspeptins in female puberty and preovulatory gonadotropin surges as revealed by a novel antagonist.

Pineda. R R; Garcia-Galiano. D D; Roseweir. A A; Romero. M M; Sanchez-Garrido. M A MA; Ruiz-Pino. F...

Scientists gave female rats a drug that blocks kisspeptin, a hormone that triggers reproductive signals. Continuous brain infusion of this blocker delayed puberty signs and stopped the normal hormone surge that leads to ovulation. A version that can cross the blood‑brain barrier also reduced the hormone spikes caused by kisspeptin when given by injection.

Utility 1
pubmed Sep 19, 2010

Anatomy of the kisspeptin neural network in mammals.

Lehman. Michael N MN; Merkley. Christina M CM; Coolen. Lique M LM; Goodman. Robert L RL

Kisspeptin is a brain chemical that helps control the release of reproductive hormones, and this paper maps where kisspeptin‑producing cells are in the brain and how they connect with each other and with GnRH neurons.

Utility 1
pubmed Aug 1, 2010

The role of kisspeptin signaling in reproduction.

d'Anglemont de Tassigny. Xavier X; Colledge. William Henry WH

Kisspeptin is a small protein that tells the brain to release hormones needed for puberty and normal reproductive function. This review explains how kisspeptin acts as a central hub, gathering many hormonal and body signals to control fertility.

Utility 1
pubmed Jul 5, 2012

First-trimester maternal serum metastin, placental growth factor and chitotriosidase levels in pre-eclampsia.

Madazli. Riza R; Bulut. Berk B; Tuten. Abdullah A; Aydin. Burcu B; Demirayak. Gökhan G; Kucur....

A study found that pregnant women who later develop pre‑eclampsia have lower levels of the peptide kisspeptin‑10 (also called metastin) and placental growth factor, and higher activity of an enzyme called chitotriosidase, already in the first trimester. These differences could help doctors spot the risk early, but the research doesn’t suggest any new treatment or supplement for the general public.